Xi'an ruixi Biological Technology Co

Home > Keywords >

Catalog	name	Description	price
R-R-4103	Taranabant racemate CAS No.701977-00-6	Taranabant racemate (MK-0364 racemate)/CAS No.701977-00-6 is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1.	price>
R-C-2404	Piribedil CAS:3605-01-4	Piribedil(Trivastal,Trivastan)is a relatively selective dopamine(D2/D3)agonist with moderate antidepressant activity.It also has α2-adrenergic(α2A/α2C)antagonist properties.	price>
R-R-4104	SCH 336 CAS No.447459-51-0	SCH 336/CAS No.447459-51-0 is a potent, selective, inverse and orally active CB2 agonist. SCH 336 inhibits BaF3/CB2 migration. SCH 336 significantly inhibits the migration of leukocytes in vivo. SCH 336 blocks ovalbumin-induced lung eosinophilia in mice.	price>
R-C-2405	SR59230A CAS:174689-39-5	SR59230A is a blood-brain barrier penetrating,potent and selective antagonist of β3-adrenergic receptor with IC50 of 40nM,408nM,and 648nM for β3,β1,and β2 receptors,respectively.	price>
R-R-4105	Tetrahydromagnolol CAS No.20601-85-8	Tetrahydromagnolol (Magnolignan)/CAS No.20601-85-8, a main metabolite of Magnolol, is a potent and selective cannabinoid CB2 receptor agonist with an EC50 of 170 nM and a Ki of 416 nM. Tetrahydromagnolol possesses 20-fold more selective for CB2 receptor than CB1 receptor. Tetrahydromagnolol is also a weak GPR55 receptor antagonist.	price>
R-R-4106	AZD1940 CAS No.881413-29-2	AZD1940/CAS No.881413-29-2 is an orally active, high affinity cannabinoid CB1/CB2 receptor agonist with pKi values of 7.93 and 9.06 for human CB1R and CB2R, respectively. AZD1940 shows a robust analgesia action.	price>
R-C-2407	Desvenlafaxine CAS:93413-62-8	Desvenlafaxine is a synthetic form of the major active metabolite of venlafaxine (sold under the brand names Effexor and Efexor).It is being targeted as the first non-hormonal based treatment for menopause.Desvenlafaxine is a synthetic phenethylamine bicyclic derivative with antidepressant activity. Desvenlafaxine is a selective reuptake inhibitor of serotonin and norepinephrine due to its high binding affinities to the pre-synaptic serotonin and norepinephrine transporters.	price>
R-R-4107	Vicasinabin CAS No.1433361-02-4	Vicasinabin (RG7774)/CAS No.1433361-02-4 is the potent agonist of cannabinoid receptor 2 (CB2). Vicasinabin has the potential for the research of human diseases including chronic pain, atherosclerosis, regulation of bone mass, neuroinflammation, and other related diseases (extracted from patent US20130116236A1).	price>
R-C-2408	Esmolol CAS:81147-92-4	Esmolol is a short acting hyperselective β-adrenergic blocker effective in blunting adrenergic response to several perioperative stimuli and so it might interfere in the effect of the anesthetic drugs on the brain.Esmolol is effective not only in attenuating intraoperative hemodynamic changes related to sympathetic overdrive but also in minimizing significant propofol and sevoflurane requirements without compromising the hemodynamic status.	price>
R-R-4108	LH21 CAS No.611207-11-5	LH-21/CAS No.611207-11-5 is a potent in vivo neutral cannabinoid CB1 receptor antagonist. LH-21 reduces food intake and body weight gain in obese Zucker rats. , and displays efficacy as a feeding inhibitor.	price>
R-C-2409	Doxazosin CAS: 74191-85-8	Doxazosin(UK 33274)is a quinazoline-derivative that selectively antagonizes postsynaptic α1-adrenergic receptors.	price>
R-R-4109	S-777469 CAS No.885496-53-7	S-777469/CAS No.885496-53-7 is a selective and orally available cannabinoid type 2 receptor (CB2) agonist with a Ki of 36 nM. S-777469 significantly suppresses compound 48/80-induced scratching behavior in mice in a dose-dependent manner. S-777469 produces its antipruritic effects by inhibiting itch signal transmission through CB2 agonism.	price>
R-C-2410	Nadolol CAS:42200-33-9	Nadolol(SQ-11725)is a non-selective and orally active β-adrenergic receptors blocker and is a substrate of organic anion transporting polypeptide 1A2(OATP1A2).Nadolol has the the potential for high blood pressure,angina pectoris and vascular headaches research.	price>
R-R-4110	2-Arachidonoylglycerol-d8 CAS No.924894-97-3	2-Arachidonoylglycerol-d8/CAS No.924894-97-3 is the deuterium labeled 2-Arachidonoylglycerol. 2-Arachidonoylglycerol is a second endogenous cannabinoid ligand in the central nervous system.	price>
R-C-2411	Betaxolol CAS:63659-18-7	Betaxolol is a selective beta1 receptor blocker used in the treatment of hypertension and glaucoma.Being selective for beta1+ receptors,it typically has fewer systemic side effects than non-selective beta-blockers,for example,not causing bronchospasm(mediated by beta2 receptors)as timolol may.Betaxolol also shows greater affininty for beta1 receptors than metoprolol.	price>
R-R-4111	NESS 0327 CAS No.494844-07-4	NESS 0327/CAS No.494844-07-4 is a cannabinoid antagonist with high selectivity for the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.	price>
R-C-2412	Carazolol CAS: 57775-29-8	Carazolol is a beta1/beta2 adrenoceptor antagonist of high potency used in the treatment of hypertension.Its affinity for the beta 3-adrenoceptor was determined in Chinese hamster ovary cells transfected with the gene of the human or the murine beta 3-adrenoceptor.Carazolol is recognized with a nanomolar affinity,which positions it among the best ligands for beta 3-adrenoceptors.	price>
R-R-4112	CB2 modulator 1 CAS No.666261-80-9	CB2 modulator 1 (compound 130)/CAS No.666261-80-9 is a potent CB2 modulator. CB2 modulator 1 has the potential for immunedisorders, inflammation, osteoporosis, renal ischemia.	price>
R-C-2413	Metoprolol CAS：51384-51-1	Metoprolol(Toprol)is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system,especially hypertension.	price>
R-R-4113	AM-6538 CAS No.1245626-00-9	AM6538/CAS No.1245626-00-9 is a long-acting, high affinity and pseudo-irreversible cannabinoid (CB) antagonist. AM6538 is a structural analog of rimonabant. AM6538 can be effectively used to evaluate the apparent efficacy of cannabinoid full and partial agonists. AM6538 may be useful in future studies that require temporary reductions in cannabinoid receptor availability. AM-6538 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>

616617618619620621 622623624625626