Xi'an ruixi Biological Technology Co

Home > Keywords >

Catalog	name	Description	price
R-R-4112	CB2 modulator 1 CAS No.666261-80-9	CB2 modulator 1 (compound 130)/CAS No.666261-80-9 is a potent CB2 modulator. CB2 modulator 1 has the potential for immunedisorders, inflammation, osteoporosis, renal ischemia.	price>
R-C-2413	Metoprolol CAS：51384-51-1	Metoprolol(Toprol)is a selective β1 receptor blocker used in treatment of several diseases of the cardiovascular system,especially hypertension.	price>
R-R-4113	AM-6538 CAS No.1245626-00-9	AM6538/CAS No.1245626-00-9 is a long-acting, high affinity and pseudo-irreversible cannabinoid (CB) antagonist. AM6538 is a structural analog of rimonabant. AM6538 can be effectively used to evaluate the apparent efficacy of cannabinoid full and partial agonists. AM6538 may be useful in future studies that require temporary reductions in cannabinoid receptor availability. AM-6538 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.	price>
R-C-2414	Atenolol CAS：29122-68-7	Atenolol((RS)-Atenolol)is a cardioselective β1-adrenergic receptor blocker,with a Ki of 697nM atβ1-adrenoceptor in guine pig left ventricle membrane.Atenolol can be used for the research of hypertension and angina pectoris.	price>
R-R-4114	CB2R antagonist 3	CB2R antagonist 3 is a selective antagonist of cannabinoid type 2 receptor (CB2R). CB2R antagonist 3 has high affinity for human CB2R and specific selectivity for CB1R. CB2R antagonist 3 can be combined with CB65 (HY-110047), the activator of CB2R. CB2R antagonist 3 effectively up-regulates the expression of anti-inflammatory cytokines and down-regulates the expression of pro-inflammatory cytokines.	price>
R-C-2415	Nicergoline CAS：27848-84-6	Nicergoline,an ergoline derivative ester of bromonicotinic acid,is a potent, selective and orally active antagonist of α1A-adrenoceptor.Nicergoline has vasodilator effects.Nicergoline also has ameliorative effects on cognitive function in mouse models of Alzheimer is disease.	price>
R-R-4115	CB1/2 agonist 3 CAS No.2772655-86-2	CB1/2 agonist 3 (compound 52)/CAS No.2772655-86-2, a potent non-selective cannabinoid ligand, is a CB1/CB2 (cannabinoid receptor) competitive agonist. CB1/2 agonist 3 acts on hCB1 and hCB2 with Ki values of 5.9 nM and 3.5 nM, respectively.	price>
R-C-2416	Mirabegron CAS： 223673-61-8	Mirabegron(formerly YM-178,trade name Myrbetriq)is a drug for the treatment of overactive bladder.Mirabegron activates the β3 adrenergic receptor in the detrusor muscle in the bladder,which leads to muscle relaxation and an increase in bladder capacity.	price>
R-R-4116	2-Arachidonoylglycerol-d5 CAS No.2522598-88-3	2-Arachidonoylglycerol-d5/CAS No.2522598-88-3 is the deuterium labeled 2-Arachidonoylglycerol. 2-Arachidonoylglycerol is a second endogenous cannabinoid ligand in the central nervous system.	price>
R-C-2417	Olodaterol (BI 1744) CAS:868049-49-4	Olodaterol(BI 1744)is a long-acting β2-adrenergic receptor agonist that is used as a component of an inhalation(Tiotropium/Olodaterol)for treating patients with chronic obstructive pulmonary disease(COPD).	price>
R-R-4117	JTE-907 CAS No.282089-49-0	JTE-907/CAS No.282089-49-0 is a highly selective, orally active CB2 receptor inverse agonist and exerts anti-inflammatory effects in vivo.	price>
R-C-2418	Guanabenz CAS:5051-62-7	Guanabenz(Acetate)(BR-750)is an alpha-2 selective adrenergic agonist used as an antihypertensive agent.	price>
R-R-4118	GP1a CAS No.511532-96-0	GP1a/CAS No.511532-96-0 is a potent agonist of cannabinoid receptor 2 (CB2). Gp1a is beneficial to skin wound healing. GP1a inhibits inflammation and fibrogenesis while promoting re-epithelialization.	price>
R-C-2419	Droxidopa CAS:23651-95-8	Droxidopa is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitters norepinephrine(noradrenaline)and epinephrine(adrenaline)and it is used to increase the concentrations of these neurotransmitters in the body and brain.Unlike norepinephrine and epinephrine themselves,droxidopa is capable of crossing the protective bloodÂ–brain barrier(BBB).	price>
R-R-4119	RVD-Hpα TFA CAS No.1431329-51-9	RVD-Hpα TFA/CAS No.1431329-51-9 is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).	price>
R-C-2420	Dexmedetomidine CAS:113775-47-6	Dexmedetomidine is notable for its ability to provide sedation without risk of respiratory depression(unlike other commonly used sedatives such as propofol, fentanyl,and midazolam)and can provide cooperative or semi-arousable sedation.	price>
R-R-4120	BML-190 CAS No.2854-32-2	BML-190(IMMA)/CAS No.2854-32-2 is a potent and selective CB2 receptor ligand (Ki values are 435 nM and > 2 μM for CB2 and CB1 respectively).	price>
R-C-2421	Pimethixene maleate CAS:13187-06-9	Pimethixene(Pimetixene)maleate,an antihistamine,anntimigraine agent and antiserotonergic compound,is a highly potent antagonist of a broad range of monoamine receptors,including a variety of serotonin receptors.	price>
R-R-4121	Auriculasin CAS No.60297-37-2	Auriculasin/CAS No.60297-37-2 is a nature product isolated from Limonium leptophyllum. Auriculasin has activity toward cannabinoid receptor type 1 (CB1) with an IC50 value of 8.92 µM.	price>
R-C-2422	Varenicline Hydrochloride CAS:230615-23-3	Varenicline Hydrochloride(CP 526555 hydrochloride)is a high affinity, selective α4β2 nicotine acetylcholine receptor(nAChR)partial agonist and full α7 nAChR agonist.Varenicline Hydrochloride is also a potent partial agonist of α6β2 nAChR in striatum of rats with a Ki value of 0.12nM.	price>

610611612613614615 616617618619620