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Catalog	name	Description	price
R-C-2202	Ramucirumab (anti-VEGFR2) CAS:947687-13-0	Ramucirumab is a human VEGFR-2 antagonist for the treatment of solid tumors. Ramucirumab is a recombinant human immunoglobulin G1 monoclonal antibody that binds to the extracellular binding domain of VEGFR-2 and prevents the binding of VEGFR ligands:VEGF-A,VEGF-C,and VEGF-D.	price>
R-R-3902	Salmeterol-d3 CAS No.497063-94-2	Salmeterol-d3/CAS No.497063-94-2 is a deuterium labeled Salmeterol. Salmeterol is a potent and selective human β2 adrenoceptor agonist. Salmeterol shows potent stimulation of cAMP accumulation in CHO cells expressing human β2, β1 and β3 adrenoceptors with pEC50s of 9.6, 6.1, and 5.9, respectively.	price>
R-C-2203	Sulfatinib CAS:1308672-74-3	Sulfatinib(HMPL-012)is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3,FGFR1 and CSF1R with IC50s of in a range of 1 to 24nM.	price>
R-R-3903	Guanoxabenz hydrochloride CAS No.23256-40-8	Guanoxabenz (Hydroxyguanabenz) hydrochloride/CAS No.23256-40-8 is an α2 adrenergic receptor agonist, with a Ki of 4000 nM and the fully activated form 40 nM for an α2A adrenoceptor.	price>
R-C-2204	Taxifolin (Dihydroquercetin) CAS:480-18-2	Taxifolin((+)-Dihydroquercetin)exhibits important anti-tyrosinase activity.Taxifolin exhibits significant inhibitory activity against collagenase with an IC50 value of 193.3μM.Taxifolin is an important natural compound with antifibrotic activity.Taxifolin is a free radical scavenger with antioxidant capacity.	price>
R-R-3904	Arbutamine CAS No.128470-16-6	Arbutamine/CAS No.128470-16-6 is a short-acting, potent and nonselective β-adrenoceptor agonist. Arbutamine stimulates cardiac β1-, tracheal β2-, and adiopocyte β3- adrenergic receptors. Arbutamine provides cardiac stress increases heart rate, cardiac contractility, and systolic blood pressure. Arbutamine can be used for cardiac stress agent .	price>
R-C-2205	SU5214 CAS: 186611-04-1	SU5214 is a potent VEGFR2 inhibitor extracted from patent US5834504A,SU5214, has IC50s of 14.8µM(FLK-1)and 36.7µM(EGFR),respectively.	price>
R-R-3905	Efaroxan hydrochloride CAS No.89197-00-2	Efaroxan hydrochloride/CAS No.89197-00-2 is a potent, selective and orally active α2-adrenoceptor antagonist, with antidiabetic activity. Efaroxan hydrochloride is a selective I1-Imidazoline receptor antagonist. Efaroxan hydrochloride can be used for the research of cardiovascular disease.	price>
R-C-2206	SU5408 CAS:15966-93-5	SU5408(VEGFR2 Kinase Inhibitor I)is a potent and cell-permeable inhibitor of VEGFR2 kinase with an IC50 of 70nM.	price>
R-R-3906	NP10679	NP10679 is a selective, pH dependent GluN2B subunit-specific N-methyl-D-aspartate (NMDA) receptor inhibitor with high oral bioavailability and good brain penetration. NP10679 inhibits GluN2B with IC50s of 23 and 142 nM at pH 6.9 and 7.6, respectively. NP10679 is a histamine H1 antagonist and a hERG channel inhibitor with IC50s of 73 and 620 nM, respectively. NP10679 is a reversible inhibitor of human liver CYP enzymes.	price>
R-C-2207	SU5205 CAS:3476-86-6	SU5205 is an inhibitor of VEGFR2 (FLK-1),with an IC50 of 9.6μM.	price>
R-R-3907	Scopine hydrochloride CAS No.85700-55-6	Scopine hydrochloride (6,7-Epoxytropine hydrochloride)/CAS No.85700-55-6 is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.	price>
R-C-2208	2-D08 CAS:144707-18-6	2-D08 is a cell permeable,mechanistically unique inhibitor of protein sumoylation.It is also inhibits Axl,IRAK4,ROS1,MLK4,GSK3β,RET,KDR and PI3Kα with IC50 values of 0.49,3.9,5.3,9.8,11,11,17 and 35nM respectively in biochemical assays.	price>
R-R-3908	Bunazosin CAS No.80755-51-7	Bunazosin/CAS No.80755-51-7 is a potent and selective α1-adrenoceptor antagonist. Bunazosin can be used for antihypertensive and ocular hypotensive research.	price>
R-C-2209	CS-2660 (JNJ-38158471) CAS:951151-97-6	CS-2660(JNJ-38158471)is a well tolerated,orally available,highly selective VEGFR-2 inhibitor with IC50 of 40 nM.CS-2660(JNJ-38158471)also inhibits closely related tyrosine kinases such as RET(c-RET)and Kit(c-Kit)with IC50 of 180nM and 500nMwhile it has no significant activity(>1 microM) against VEGFR-1 and VEGFR-3.	price>
R-R-3909	Salbutamol-d3 CAS No.1219798-60-3	Salbutamol-d3/CAS No.1219798-60-3 is the deuterium labeled Salbutamol. Salbutamol is a short-acting β2-adrenergic receptor agonist used for the relief of bronchospasm in conditions such as asthma and chronic obstructive pulmonary disease (COPD).	price>
R-C-2210	Ningetinib CAS:1394820-69-9	Ningetinib is a potent,orally bioavailable small molecule tyrosine kinase inhibitor(TKI)with IC50s of 6.7,1.9 and<1.0nM for c-Met,VEGFR2 and Axl,respectively.	price>
R-R-3910	Midaglizole CAS No.66529-17-7	Midaglizole ((±)-DG5128 free base, DG5128 free base)/CAS No.66529-17-7 is a potent α2-adrenoceptor antagonist. Midaglizole is a hypoglycemic agent. Midaglizole increases blood pressure and reduces blood glucose levels in vivo.	price>
R-C-2211	CZC-8004 CAS:916603-07-1	CZC-8004 is a pan-kinase inhibitor and binds a range of tyrosine kinases, including ABL kinase.	price>
R-R-3911	ICI 89406 CAS No.53671-71-9	ICI 89406/CAS No.53671-71-9 is a selective β1 adrenergic receptor antagonist amenable to labelling with positron emitters, for PET.	price>

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