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Catalog | name | Description | price |
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R-C-2364 | Closantel CAS:57808-65-8 | Closantel is a halogenated salicylanilide with a potent anti-parasitic activity.Closantel is a potent and highly specific Onchocerca volvulus chitinase(OvCHT1)inhibitor with an IC50 of 1.6μM and a Ki of 468nM.Closantel inhibits the O.volvulus L3 to L4 molt of developing. | price> |
R-R-4064 | PD 168368 CAS No.204066-82-0 | PD 168368/CAS No.204066-82-0 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15–45 nM. PD 168368 is neuromedin B receptor (NMBR; IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively. | price> |
R-C-2365 | Ftaxilide CAS:19368-18-4 | Ftaxilide is a bioactive chemical. | price> |
R-R-4065 | Kuwanon G CAS No.75629-19-5 | Kuwanon G/CAS No.75629-19-5 is a flavonoid isolated from Morus alba, acts as a bombesin receptor antagonist, with potential antimicrobial activity. | price> |
R-C-2366 | Pasiniazid CAS:2066-89-9 | Pasiniazid is a biochemical used in the treatment of tuberculosis. | price> |
R-R-4066 | Kuwanon H CAS No.76472-87-2 | Kuwanon H/CAS No.76472-87-2 is a flavonoid isolated from Morus alba, which acts as a potent non-peptide bombesin receptor antagonist. Kuwanon H selectively inhibits binding of gastrin releasing peptide CRP to GRP-preferring recepotr, with a Ki value of 290 nM in cells. | price> |
R-C-2367 | BTZ043 Racemate CAS:957217-65-1 | BTZ043 Racemate(BTZ10526038)is the racemate of BTZ043.BTZ043 is an inhibitor of decaprenyl-phosphoribose-epimerase(DprE1),and the antimicrobial activity of BTZ043 is more potent than BTZ043 Racemate. | price> |
R-R-4067 | Bradykinin CAS No.58-82-2 | Bradykinin/CAS No.58-82-2 is an active peptide that is generated by the kallikrein-kinin system. It is a inflammatory mediator and also recognized as a neuromediator and regulator of several vascular and renal functions. | price> |
R-C-2368 | Tigecycline (GAR-936) CAS:220620-09-7 | Tigecycline(GAR-936)is bacteriostatic and is a protein synthesis inhibitor by binding to the 30S ribosomal subunit of bacteria and thereby blocking entry of Aminoacyl-tRNA into the A site of the ribosome during prokaryotic translation. Tigecycline induces autophagy by downregulating the PI3K-AKT-mTOR pathway. | price> |
R-R-4068 | Icatibant CAS No.130308-48-4 | Icatibant (HOE-140)/CAS No.130308-48-4 is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively. | price> |
R-C-2369 | Rifabutin (LM427) CAS:72559-06-9 | Rifabutin(Ansamycin)is a semisynthetic ansamycin antibiotic with potent antimycobacterial properties.Rifabutin inhibits DNA-dependent RNA polymerase. | price> |
R-R-4069 | Icatibant acetate CAS No.138614-30-9 | Icatibant acetate (HOE-140 acetate)/CAS No.138614-30-9 is a potent and specific peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively. | price> |
R-C-2370 | Biapenem CAS:120410-24-4 | Biapenem(CLI 86815;L 627;LJC10627)a parenteral carbapenem antibacterial agent with a broad spectrum. | price> |
R-R-4070 | Lobradimil CAS No.159768-75-9 | Lobradimil (RMP 7)/CAS No.159768-75-9, a synthetic bradykinin analog, is a potent and selective bradykinin B2 receptor agonist (Ki: 0.54 nM). Lobradimil increases the permeability of the BBB. Lobradimil can be used in the research of brain tumors. | price> |
R-C-2371 | Teicoplanin CAS:61036-62-2 | Teicoplanin is a semisynthetic glycopeptide antibiotic used in the prophylaxis and treatment of serious infections caused by Gram-positive bacteria,including Methicillin-resistant Staphylococcus aureus and Enterococcus faecalis. | price> |
R-R-4071 | R715 CAS No.185052-09-9 | R715/CAS No.185052-09-9 is a selective bradykinin B1 receptor antagonist. R715 significantly attenuates the hyperalgesic effect developed in Streptozotocin(HY-13753)-diabetic mice. | price> |
R-C-2372 | Aztreonam CAS:78110-38-0 | Aztreonam(SQ-26,776)is a synthetic monocyclic beta-lactam antibiotic,which has a very high affinity for penicillin-binding protein 3(PBP-3). | price> |
R-R-4072 | MEN 11270 CAS No.235082-52-7 | MEN 11270/CAS No.235082-52-7, a cyclic decapeptide, is a B2 kinin receptor antagonist. MEN 11270 bound with high-affinity to the B2 kinin receptor constitutively expressed by WI38 human fibroblasts, inhibiting 3H-bradykinin (BK) with a pKi value of 10.3. | price> |
R-C-2373 | Cefditoren Pivoxil CAS:117467-28-4 | Cefditoren pivoxil is a new-third generation cephalosporin antibiotic that has a broad spectrum of activity against Gram-positive and Gram-negative bacteria,including common respiratory and skin pathogens. | price> |
R-C-3033 | CAY10505 CAS:1218777-13-9 | CAY10505 is a potent inhibitor of PI3K, selectively inhibiting the γ isoform (IC50 = 30 nM) better than the α, β, and δ isoforms (IC50 = 0.94, 20, and 20 μM, respectively).Only for scientific research, not for human body. | price> |