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Catalog	name	Description	price
R-R-4024	Telmisartan-d3 CAS No.1189889-44-8	Telmisartan-d3/CAS No.1189889-44-8 is the deuterium labeled Telmisartan. Telmisartan is a potent, long lasting antagonist of angiotensin II type 1 receptor (AT1), selectively inhibiting the binding of 125I-AngII to AT1 receptors with IC50 of 9.2 nM.	price>
R-C-2325	Protopine CAS:130-86-9	Protopine(Corydinine,Fumarine,Biflorine,Macleyine),an alkaloid present in different plants,has been shown to exhibit a number of activities,such as inhibition of calcium influx through both voltage and receptor-operated channels and inhibition of rabbit blood platelet aggregation.It also possesses anti-cholinergic and anti-histaminic as well as anti-bacterial activities.	price>
R-R-4025	Eprosartan mesylate CAS No.144143-96-4	Eprosartan mesylate (SKF-108566J)/CAS No.144143-96-4 is a selective, competitive, nonpeptid and orally active angiotensin II receptor antagonist, used as an antihypertensive. Eprosartan mesylate binds angiotensin II receptor with IC50s of 9.2 nM and 3.9 nM in rat and human adrenal cortical membranes, respectively.	price>
R-C-2326	Trimethadione CAS:127-48-0	Trimethadione(3,5,5,-Trimethyloxazolidine-2,4-dione)is an oxazolidinedione anticonvulsant agent widely used against absences seizures.Trimethadione also is a T-type calcium channel blocker which has antihyperalgesic effects.	price>
R-R-4026	Candesartan-d4 CAS No.1346604-70-3	Candesartan-d4/CAS No.1346604-70-3 is the deuterium labeled Candesartan, which is an angiotensin II receptor antagonist.	price>
R-C-2327	SN-6 CAS: 415697-08-4	SN-6 is a selective Na+/Ca2+ exchanger(NCX)inhibitor.SN-6 inhibits NCX1,NCX2, and NCX3 with IC50 of 2.9μM,16μM and 8.6μM, respectively.SN-6 abolishes acetylcholine(ACh)-induced vasodilation.	price>
R-R-4027	Olmesartan lactone impurity CAS No.849206-43-5	Olmesartan lactone impurity/CAS No.849206-43-5 is a cyclic ester impurity of Olmesartan. Olmesartan is an angiotensin II receptor (AT1R) antagonist and has the potential for high blood pressure study.	price>
R-C-2328	Pinaverium bromide CAS:53251-94-8	Pinaverium bromide is an L-type calcium channel blocker with selectivity for the gastrointestinal tract,effectively relieves pain,diarrhea and intestinal discomfort,provides good therapeutic efficacies without significant adverse effects on Irritable bowel syndrome(IBS)patients.	price>
R-R-4028	Losartan-d4 (carboxylic acid) CAS No.1246820-62-1	Losartan-d4 (carboxylic acid)/CAS No.1246820-62-1 is the deuterium labeled Losartan (EXP-3174), which is an angiotensin II receptor antagonist.	price>
R-C-2329	Strontium Ranelate CAS:135459-87-9	Strontium Ranelate(S12911)is an antiosteoporotic agent that acts by reducing bone resorption and promoting bone formation,thereby inducing a positive bone balance.Strontium Ranelate also can activate the calcium-sensing receptor (CaSR)in non skeletal cells,resulting in the activation of inositol 1,4,5-triphosphate production and mitogen-activated protein kinase signaling.	price>
R-R-4029	Angiotensin II (5-8), human	Angiotensin II (5-8), human is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II. Angiotensin II binds the AT II type 1 (AT1) receptor, stimulating GPCRs in vascular smooth muscle cells and increasing intracellular Ca2+ levels. Angiotensin II also acts at the Na+/H+ exchanger in the proximal tubules of the kidney.	price>
R-C-2330	Bay K 8644 CAS:71145-03-4	Bay K 8644,a dihydropyridine compound,is a specific L-type Ca2+channel agonist.Bay K 8644 increases Ca2+ influx through sarcolemmal Ca2+channels by increasing the open time of the channel.	price>
R-R-4030	Losartan-d4 CAS No.1030937-27-9	Losartan-d4/CAS No.1030937-27-9 is the deuterium labeled Losartan. Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM.	price>
R-C-2331	Salbutamol CAS:18559-94-9	Salbutamol(Albuterol)is a short-acting,selective beta2-adrenergic receptor agonist used to treat or prevent bronchospasm in patients with asthma, bronchitis,emphysema,and other lung diseases.	price>
R-R-4031	trans-Tranilast CAS No.70806-55-2	trans-Tranilast (trans-MK-341)/CAS No.70806-55-2 is an antiallergic drug, used to treat bronchial asthma, allergic rhinitis and atopic dermatitis.	price>
R-C-2332	Brimonidine CAS:59803-98-4	Brimonidine is a drug used as eye drops under the brand names Alphagan and Alphagan-P to treat open-angle glaucoma or ocular hypertension.	price>
R-R-4032	Valsartan-d9 CAS No.1089736-73-1	Valsartan-d9/CAS No.1089736-73-1 is deuterium labeled valsartan. Valsartan is an angiotensin II receptor antagonist and has the potential for high blood pressure and heart failure research.	price>
R-C-2333	Synephrine CAS:94-07-5	Synephrine(Oxedrine),an alkaloid,is an α-adrenergic and β-adrenergic agonist derived from the Citrus aurantium.Synephrine is a sympathomimetic compound and can be used for weight loss.	price>
R-R-4033	TD-0212 TFA CAS No.1073549-11-7	TD-0212 TFA/CAS No.1073549-11-7 is an orally active dual pharmacology angiotensin II type 1 receptor (AT1) antagonist and neprilysin (NEP) inhibitor, with a pKi of 8.9 for AT1 and a pIC50 of 9.2 for NEP.	price>
R-C-2334	Indacaterol CAS:312753-06-3	Indacaterol(Onbrez;Arcapta)is an ultra-long-acting β-adrenoceptor agonist.	price>

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