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Catalog	name	Description	price
R-C-1830	Etofenamate CAS：30544-47-9	Etofenamate is a nonsteroidal anti-inflammatory drug(NSAID)used for the treatment of joint and muscular pain.	price>
R-R-3530	MRS 1523 CAS No.212329-37-8	MRS 1523/CAS No.212329-37-8 is a potent and selective adenosine A3 receptor antagonist with Ki values of 18.9 nM and 113 nM for human and rat A3 receptors, respectively. In rat this corresponds to selectivities of 140- and 18-fold vs A1 and A2A receptors, respectively. MRS 1523 can exert antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons.	price>
R-GNG0405-X	Polysaccharide modified gold nanorods（GNRs）	Polysaccharide modified gold nanorods(GNRs),cas7440-57-5,Glucose,Maltose and Dextran is optional.	price>
R-C-1831	Hydroxyfasudil hydrochloride(HA-1100) CAS:155558-32-0	Hydroxyfasudil hydrochloride is a ROCK inhibitor,with IC50s of 0.73 and 0.72 μM for ROCK1 and ROCK2,respectively.	price>
R-R-3531	CGS 15943 CAS No.104615-18-1	CGS 15943/CAS No.104615-18-1 is an orally bioavailable non-xanthine Adenosine Receptor antagonist. Its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM in transfected CHO cells, respectively.	price>
R-GN010005	Gold Nanorods, Streptavidin function	Gold Nanorods, Streptavidin function,cas7440-57-5	price>
R-GNPE0401-X	Gold nanorods, AuNRs-PEG-Silane	Gold nanorods, polyethylene glycol silane function,cas7440-57-5	price>
R-C-1832	MG-132 CAS:1211877-36-9	MG132(Z-Leu-Leu-Leu-al)is a potent cell-permeable proteasome and calpain inhibitor with IC50s of 0.1μM and 1.2μM for the inhibition of proteasome and calpain,respectively.MG132 activates autophagy and induces apoptosis in tumor cells.	price>
R-R-3532	Tonapofylline CAS No.340021-17-2	Tonapofylline (BG 9928)/CAS No.340021-17-2 is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure.	price>
R-GNPLGA0201-x	Gold nanorods,AuNRs-PEG-PLGA	Gold nanorods, polyethylene glycol and poly(lactic-co-glycolic acid) function, cas7440-57-5	price>
R-C-1833	UNC3866 CAS:1872382-47-2	UNC3866 is a potent antagonist of the methyllysine(Kme)reading function of the Polycomb CBX and CDY families of chromodomains.UNC3866 binds the chromodomains of CBX4 and CBX7 most potently,with a K(d)of∼100nM for each,and is 6- to 18-fold selective as compared to seven other CBX and CDY chromodomains.	price>
R-R-3533	Rolofylline CAS No.136199-02-5	Rolofylline (KW-3902)/CAS No.136199-02-5 is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. Rolofylline is metabolized primarily to the pharmacologically active M1-trans and M1-cis metabolites by cytochrome P450 (CYP450). Rolofylline is alleviating the presynaptic dysfunction and restores neuronal activity as well as dendritic spine levels in vitro, is an interesting candidate to combat the hypometabolism and neuronal dysfunction associated with Tau-induced neurodegenerative diseases.	price>
R-GNPLA0501-X	Gold nanorods, AuNRs-PEG-PLA	Gold Nanoparticles,polyethylene glycol poly(L-lactide) function,cas7440-57-5	price>
R-C-1834	BV6 CAS:1001600-56-1	BV6 is an inhibitor of apoptosis(IAP)proteins.It acts by promoting glioblastoma cancer stem-like cell differentiation by activating NF-κB.	price>
R-R-3534	Taminadenant CAS No.1337962-47-6	Taminadenant (NIR178; PBF509)/CAS No.1337962-47-6 is a highly potent and orally active adenosine A2A receptor (A2AR) antagonist. Taminadenant can antagonize A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 nM and 8.2 nM, respectively. Taminadenant reverses motor impairments in several rat models of movement disorders, including catalepsy, tremor, and hemiparkinsonism. Taminadenant can also inhibit tumor growth when combined with Spartalizumab (HY-P9972). Taminadenant reactivate the antitumor immune response.	price>
R-GNPCL0401-X	Gold nanorods, AuNRs-PEG-PCL	Gold nanorods, polyethylene glycol poly(caprolactone) function, cas7440-57-5	price>
R-C-1835	MM-102 CAS:1417329-24-8	MM-102(HMTase Inhibitor IX)is a high-affinity peptidomimetic MLL1 inhibitor with IC50 of 0.4μM in a cell-free assay.	price>
R-R-3535	Doxofylline CAS No.69975-86-6	Doxofylline/CAS No.69975-86-6 is an orally active PDE IV inhibitor and A1AR antagonist. Doxofylline reduces inflammation in epithelial cells via inhibiting mitochondrial ROS production and amelioration of multiple cellular pathways (NLRP3-TXNIP inflammasome activation). Doxophylline can be used in studies of asthma, chronic obstructive pulmonary disease, and bronchospasm.	price>
R-GNPEI0405-X	Gold nanorods, AuNRs-PEG-PEI	Gold nanorods, polyethylene glycol polyetherimide function, cas7440-57-5	price>
R-C-1836	ULM-1(MDK7526HCL) CAS:228544-65-8	VULM-1457 is an Acyl-CoA cholesterol acyltransferase(ACAT)inhibitor.	price>

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