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Catalog	name	Description	price
R-C-1646	Lys05 CAS:1391426-22-4	Lys05 is a potent lysosomal autophagy inhibitor.Lys05 is a previously undescribed dimeric chloroquine which more potently accumulates in the lysosome and blocks autophagy compared with HCQ.	price>
R-R-3346	(S)-Amisulpride CAS No.71675-92-8	(S)-Amisulpride (Esamisulpride)/CAS No.71675-92-8 is a potent dopamine D2/D3 receptor antagonist. (S)-Amisulpride is an antagonist at the 5-HT7 receptor with a KI of 900 nM. (S)-Amisulpride has antipsychotic and antidepressant effects.	price>
R-C-1647	Importazole CAS:662163-81-7	Importazole is a small molecule inhibitor of the transport receptor importin-β (Karyopherin beta)specifically blocking importin-β-mediated nuclear import. Importazole induces apoptosis and inhibits tumor growth.	price>
R-R-3347	SB228357 CAS No.181629-93-6	SB228357/CAS No.181629-93-6 is a selective, potent and orall active 5-HT2C/2B receptor antagonist with pKi values of 6.9, 8.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. SB228357 has antidepressant/anxiolytic effects.	price>
R-C-1648	Miransertib (ARQ-092) CAS:1313881-70-7	Miransertib(ARQ-092)is a potent,selective and orally bioavailable allosteric inhibitor of Akt with IC50s of 2.7nM,14 nM and 8.1nM for Akt1,Akt2,Akt3.	price>
R-R-3348	SB-200646A CAS No.143797-62-0	SB-200646A/CAS No.143797-62-0 is the first selective 5-HT2B/2C over 5-HT2A receptor antagonist with pKi values of 7.5, 6.9 and 5.2 for 5-HT2B, 5-HT2C and 5-HT2A, respectively. SB-200646A is orally active and has electrophysiological and anxiolytic properties in vivo.	price>
R-R-3349	PU02 CAS No.313984-77-9	PU02/CAS No.313984-77-9, a derivative of 6-MP (HY-13677), is a negative allosteric modulator (NAM) of 5-HT3 receptor, with IC50 values of 0.36 and 0.73 μM in HEK293 cells transfected with human 5-HT3A and 5-HT3AB receptors respectively.	price>
R-C-1649	SKF96365.HCl CAS:130495-35-1	SKF-96365 hydrochloride is a potent TRP channel blocker and a store-operated Ca2+ entry(SOCE)inhibitor.SKF-96365 hydrochloride significantly inhibits hERG, hKCNQ1/hKCNE1,hKir2.1 and hKv4.3 current,and significantly prolongs the QTc interval in isolated guinea pig hearts.SKF-96365 hydrochloride exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal cancer cells.	price>
R-C-1650	AR-M1000390 HCl CAS:209808-47-9	AR-M1000390(ARM-390)is a nonpeptidic δ receptor selective agonist.	price>
R-R-3350	Alniditan dihydrochloride CAS No.155428-00-5	Alniditan (Alnitidan) dihydrochloride/CAS No.155428-00-5 is a potent 5-HT1B and 5-HT1D receptors agonist, with IC50s of 1.7 nM and 1.3 nM for h5-HT1B and h5-HT1D receptors in HEK 293 cells, respectively. Alniditan dihydrochloride has migraine-preventive effects.	price>
R-C-1651	nicainoprol CAS：76252-06-7	Nicainoprol is a fast-sodium-channel blocking drug,which is a potent antiarrhythmic agent.	price>
R-R-3351	Tedatioxetine hydrobromide CAS No.960151-65-9	Tedatioxetine (Lu AA24530) hydrobromide/CAS No.960151-65-9 acts as a serotonin and norepinephrine (NE)-preferring triple reuptake inhibitor (TRI) and 5-HT2A, 5-HT2C, 5-HT3 and α1A-adrenergic receptor antagonist.	price>
R-C-1652	DAA1106 CAS：220551-92-8	DAA1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR),as a potent and selective agonist at the peripheral benzodiazepine receptor.	price>
R-R-3352	Naluzotan CAS No.740873-06-7	Naluzotan/CAS No.740873-06-7 is a novel, potent, and selective amidosulfonamide 5-HT1A agonist with IC50 and Ki of appr 20 nM and 5.1 nM, used for the treatment of anxiety and depression; Also a weak hERG K+ channel blocker, with IC50 of 3800 nM.	price>
R-C-1653	Eptapirone (F11440) CAS：179756-58-2	Eptapirone(F11440)is a potent,selective,high efficacy 5-HT1A receptor agonist with marked anxiolytic and antidepressant potential.	price>
R-R-3353	Velusetrag hydrochloride CAS No.866933-51-9	Velusetrag (TD-5108) hydrochloride/CAS No.866933-51-9 is an orally active, potent and selective agonist of serotonin 5-HT4 receptor (5-HT4R), with a pKi of 7.7. Velusetrag hydrochloride exhibits no affinity (Ki>10 μM) for 5-HT2A and 5-HT2B receptors.	price>
R-C-1654	Orexin 2 Receptor Agonist CAS：1796565-52-0	Orexin 2 Receptor Agonist is a potent(EC50 on OX2R is 23nM)and OX2R-selective (OX1R/OX2R EC50 ratio is 70) agonist.	price>
R-R-3354	Aripiprazole-d8 CAS No.1089115-06-9	Aripiprazole-d8/CAS No.1089115-06-9 is the deuterium labeled Aripiprazole, which is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.	price>
R-C-1655	piperoxan.HCl CAS: 135-87-5	Piperoxan hydrochloride(Benodaine,Fourneau 933,F933,DL-Piperoxan)is an antagonist of α2(alpha 2)adrenoceptor.	price>
R-M-G25	Carbon Nanotube Aerogel	Carbon nanotube Aerogel/Carbon nanotubes(CNT) Aerogel/CNT Aerogel is a kind of carbon nanotube with dispersion properties. This paper prepared carbon nanotube aerogel through independent research and development of experimental equipment, and prepared carbon nanotube aerogel/natural rubber composite through traditional processes. Material, the mechanical properties and thermal conductivity of the composite material were studied. The results proved that the tensile strength, tear strength and thermal conductivity of the composite material were improved by 47%, 52% and 49.9 respectively compared with the carbon black/natural rubber composite material. %, while revealing the good dispersion properties of carbon nanotube airgel and its broad application prospects.	price>

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