Prexasertib dimesylate CAS No.1234015-58-7
Prexasertib dimesylate CAS No.1234015-58-7
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-1442 | 25mg | 340.00 | + Add to cart |
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R-R-1442 | 50mg | 540.00 | + Add to cart |
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Product description
Prexasertib dimesylate (LY2606368 dimesylate)/CAS No.1234015-58-7 is a selective, ATP-competitive second-generation checkpoint kinase 1 (CHK1) inhibitor with a Ki of 0.9 nM and an IC50 of <1 nM. Prexasertib dimesylate inhibits CHK2 (IC50=8 nM) and RSK1 (IC50=9 nM). Prexasertib dimesylate causes double-stranded DNA breakage and replication catastrophe resulting in apoptosis. Prexasertib dimesylate shows potent anti-tumor activity.
Appearance | N/A |
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Molecular Weight | 557.60 |
Purity | >90% |
CAS | 1234015-58-7 |
Formula | C20H27N7O8S2 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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