LY2801653 CAS:1206799-15-6
LY2801653
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-C-1683 | 50mg | 425.00 | + Add to cart |
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R-C-1683 | 100mg | 625.00 | + Add to cart |
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R-C-1683 | 200mg | 900.00 | + Add to cart |
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Product description
Merestinib(LY2801653)is a type-II ATP competitive,slow-off inhibitor of Met(c-Met)tyrosine kinase with a dissociation constant(Ki)of 2 nM, a pharmacodynamic residence time(Koff)of 0.00132 min(-1)and t1/2 of 525 min.Merestinib (LY2801653) also inhibits MST1R,AXL,ROS1,MKNK1/2, FLT3,MERTK,DDR1 and DDR2 with IC50 of 11 nM,2nM,23nM,7nM,7nM,10 nM,0.1nM and 7nM,respectively.
Appearance | N/A |
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Molecular Weight | N/A |
purity | >95% |
PDI by GPC | <1.5 |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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