GPS1573 Peptide

Catalog #	Pkg Size	Price(USD)	Quantity	Buy this product
R-M-1340	1mg	156.00	- +	+ Add to cart

Product description

GPS1573 is a newly described potent and dose-dependent peptide antagonist of ACTH-stimulated melanocortin type 2 receptor (MC2R) activity in vitro (IC50 = 66 nM). GPS1573 antagonizes MC4R with IC50 of 950 nM, therefore showing selectivity for MC2R. The binding of ACTH to MC2R regulates steroidogenesis leading to metabolic diseases such as Cushing disease in patients with pituitary dysfunctions.

Appearance	N/A
Molecular weight	N/A
Purity	>90%
Solubility	N/A
Synonyms	GPS1573; MC2R antagonist; Adrenocorticotropic hormone receptor antagonist
Sequence	H-Nle-Pro-(D-Phe)-Arg-(D-Trp)-Phe-Lys-Ala-Val-Gly-Lys-Lys-Arg-Arg-NH2 or H-Nle-PfRwFKAVGKKRR-NH2
Molecular Formula	C86H139N27O16
Storage	-20℃,protected from light and moisture
Transportation	4-25℃ temperature for up to 2 weeks
Stability	1 year

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msds of GPS1573 Peptide