CSRM617 hydrochloride CAS No.1353749-74-2
CSRM617 hydrochloride CAS No.1353749-74-2
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-1510 | 5mg | 380.00 | + Add to cart |
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R-R-1510 | 10mg | 640.00 | + Add to cart |
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Product description
CSRM617 hydrochloride/CAS No.1353749-74-2 is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2, a master regulator of androgen receptor) with a Kd of 7.43 uM in SPR assays, binding to OC2-HOX domain directly. CSRM617 hydrochloride induces apoptosis by appearance of cleaved Caspase-3 and PARP. CSRM617 hydrochloride is well tolerated in the prostate cancer mouse model.
Appearance | N/A |
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Molecular Weight | 291.69 |
Purity | >90% |
CAS | 1353749-74-2 |
Formula | C10H14ClN3O5 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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