A-192621 CAS No.195529-54-5
A-192621 CAS No.195529-54-5
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-R-1962 | 5mg | 280.00 | + Add to cart |
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R-R-1962 | 10mg | 460.00 | + Add to cart |
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Product description
A-192621/CAS No.195529-54-5 is a potent, nonpeptide, orally active and selective endothelin B (ETB) receptor antagonist with an IC50 of 4.5 nM and a Ki of 8.8 nM. The selectivity of A-192621 is 636-fold higher than ETA (IC50 of 4280 nM and Ki of 5600 nM). A-192621 promotes apoptosis in PASMCs. A-192621 alos causes elevation of arterial blood pressure and an elevation in the plasma ET-1 level.
Appearance | N/A |
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Molecular Weight | 558.66 |
Purity | >90% |
CAS | 195529-54-5 |
Formula | C33H38N2O6 |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 2 weeks |
Stability | 1 year |
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